Search Result "trypanocidal effects"


Research Article

Evaluation of Trypanocidal and Antioxidant Activities of a Selected Series of 3-amidocoumarins

Journal: Medicinal Chemistry
Volume: 14 Issue: 6 Year: 2018 Page: 573-584
Author(s): Mauricio Moncada-Basualto,Michel Lapier,Juan Diego Maya,Betty Matsuhiro,Claudio Olea-Azar,Giovanna L. Delogu,Eugenio Uriarte,Lourdes Santana,Maria Joao Matose

Review Article

Lipophilic Guanylhydrazone Analogues as Promising Trypanocidal Agents: An Extended SAR Study

Journal: Current Pharmaceutical Design
Volume: 26 Issue: 8 Year: 2020 Page: 838-866
Author(s): Vasiliki Pardali,Erofili Giannakopoulou,Dimitrios-Ilias Balourdas,Vassilios Myrianthopoulos,Martin C. Taylor,Marina Šekutor,Kata Mlinarić-Majerski,John M. Kelly,Grigoris Zoidis

Natural Products as Trypanocidal, Antileishmanial and Antimalarial Drugs

Journal: Current Topics in Medicinal Chemistry
Volume: 2 Issue: 1 Year: 2002 Page: 1215-1237
Author(s): Alain Fournet, Victoria Munoz

Trypanocidal Activity of Nitroaromatic Prodrugs: Current Treatments and Future Perspectives

Journal: Current Topics in Medicinal Chemistry
Volume: 11 Issue: 1 Year: 2011 Page: 2072-2084
Author(s): Shane R. Wilkinson, Christopher Bot, John M. Kelly, Belinda S. Hall

In Silico Study of Structural and Geometrical Requirements of Natural Sesquiterpene Lactones with Trypanocidal Activity

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 13 Issue: 1 Year: 2013 Page: 1407-1414
Author(s): L. Fabian, V. Sulsen, F. Frank, S. Cazorla, E. Malchiodi, V. Martino, E. Lizarraga, C. Catalan, A. Moglioni, L. Muschietti, L. Finkielsztein

Research Article

Synthesis of New Thiosemicarbazones and Semicarbazones Containing the 1,2,3-1H-triazole-isatin Scaffold: Trypanocidal, Cytotoxicity, Electrochemical Assays, and Molecular Docking

Journal: Medicinal Chemistry
Volume: 15 Issue: 3 Year: 2019 Page: 240-256
Author(s): Bianca N. M. Silva,Policarpo A. Sales,Alvaro J. Romanha,Silvane M. F. Murta,Camilo H. S. Lima,Magaly G. Albuquerque,Eliane D'Elia,Jose G. de Aquino,Vitor F. Ferreira,Fernando C. Silva,Angelo C. Pinto,Barbara V. Silva

Natural and Synthetic Naphthoquinones Active Against Trypanosoma Cruzi: An Initial Step Towards New Drugs for Chagas Disease

Journal: Current Medicinal Chemistry
Volume: 18 Issue: 1 Year: 2011 Page: 144-161
Author(s): Cristian O. Salas, Mario Faundez, Antonio Morello, Juan Diego Maya, Ricardo A. Tapia

Synthesis and Trypanocidal Evaluation of News 5-[N-(3-(5-Substituted)- 1,3,4-Thiadiazolyl)]Amino-1-Methyl-4-Nitroimidazoles

Journal: Letters in Drug Design & Discovery
Volume: 3 Issue: 2 Year: 2006 Page: 98-101
Author(s): A. S. Carvalho, D. Gibaldi, A. C. Pinto, M. Bozza, N. Boechat

General Research Article

New 4-nitro-imidazole-N-glycinyl-hydrazones Designed as TrypanocidalAnalogues of Benznidazole

Journal: Letters in Drug Design & Discovery
Volume: 20 Issue: 4 Year: 2023 Page: 488-497
Author(s): Juliana M. Chaves Barbosa,James L. Wardell,John N. Low,Solange M.S.V. Wardell,Samir Aquino Carvalho,Carlos Alberto Manssour Fraga

Trypanosome RNA Polymerases and Transcription Factors: Sensible Trypanocidal Drug Targets?

Journal: Current Drug Targets
Volume: 9 Issue: 1 Year: 2008 Page: 979-996
Author(s): Luc Vanhamme

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